Rolapitant

  • CAS: 552292-08-7
  • MDL:
  • Product number:QC-11703
  • Molecular formula: C25H26F6N2O2
  • Purity: 98.2%
  • MW: 500.48
Size Price Stock
25mg $680 in stock
100mg $1680 in stock
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Brief Description

Rolapitant, also known as SCH-619734, is a selective, bioavailable, CNS penetrant neurokinin NK1 receptor antagonist that shows behavioral effects in animals models of emesis. In vitro studies indicate that rolapitant has a high affinity for the human NK1 receptor of 0.66 nM and high selectivity over the human NK2 and NK3 subtypes of >1000-fold. Rolapitant is a functionally competitive antagonist, as measured by calcium efflux, with a calculated Kb of 0.17 nM.

Solubility

DMSO

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Formula Weight:

Flash point

Storage conditions

Store at -20°C 2 years

Appearance:

All CEG Chemical products are intended for laboratory research use only.

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